TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 74nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 82nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 105nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 184nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 248nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 265nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 308nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 460nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 561nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 644nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 647nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 696nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 770nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 851nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 1.16E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 1.37E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 2.02E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 5.51E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 1.36E+4nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 1.46E+4nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: >4.00E+4nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 1.30E+5nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 1.60E+5nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 1.73E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 2.03E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 2.40E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair